WHAT IS EXEMESTANE?
Exemestane, also known as Aromasin, is an Aromatase Inhibitor (AI) and is a class of drug commonly used for the treatment of breast cancer in women and gynecomastia in men. They have also been adopted by bodybuilders, who use these drugs off-label for the purpose of preventing excess estrogen levels during anabolic steroid cycles.
Exemestane is popularly used as an “estrogen blocker” which we will dig into its benefits, side-effects, results, and more below!
Manufactured by Pfizer circa 1993. It was revealed in The Mammary Prevention Trial-.3 (MAP.3) led by Canada’s NCIC Clinical Trials Group [R].
The FDA approved use of Exemestane under the brand name, Aromasin, in 1999 [R].
We’ll take a dive into the benefits, side-effects, and dosing protocol of Exemestane and allow you to make the informed decision if it’s right for your research.
HOW TO BUY EXEMESTANE
Exemestane is most commonly a prescription drug.
You can find high-quality, 3rd-party purity-tested Amino Asylum Exemestane by clicking in the link below. Use code ENHANCED20 to save 20%!
HOW DOES EXEMESTANE WORK?
Exemestane is an Aromatase Inhibitor (AI) that first is absorbed by the guy and passes through the liver enzyme CYP3A4. Once metabolized, Exemestane mobilizes to the Aromatase Enzymes or CYP19A1 and binds irreversibly, causing inactivation of the enzyme known as suicide inhibition; another name for this type of AI is called a suicidal aromatase inhibitor [R].
EXMESTANE PROS & CONS IN A NUTSHELL
- PREVENTS GYNECOMASTIA
- INCREASES TESTOSTERONE
- LOWERS ESTROGEN LEVELS
- WILL CAUSE DYSLIPIDEMIA
- MAY CRASH ESTROGEN LEVELS
- HOT FLASHES
- JOINT PAIN*
*If you’re at risk of bone fractures or have weak bones, check with your doctor before taking Exemestane.
The clinical research behind Exemestane is quite extensive. We’ve been able to compile a semi-exhaustive list of the literature behind many of these benefits and side-effects.
REDUCES ESTROGEN LEVELS
Unfortunately, Exemestane is not without side-effects and comes down to the user dosing the drug properly, under a doctor’s supervision, and with proper bloodwork results.
DECREASING BONE DENSITY
EXEMESTANE AND HIGH CHOLESTEROL
- Hot flashes
- Increased sweating
- swelling of hands or feet
- tightness in chest
HOW TO AVOID & REVERSE SIDE-EFFECTS
- Do not take Exemestane if you have osteoporosis
- Do not exceed the recommended dose of Exemestane (12.5mg)
- Do supplement with Vitamin D3, Calcium, and Potassium
- Stack a SARM, like MK-2866, to increase bone mineral density
- High Testosterone conversion needs to be in effect from the AAS you’re using
EXEMESTANE DOSAGE FOR BODYBUILDING
Bodybuilders use anywhere from 6.25mg to 25mg of Exemestane at a time but the minimum effective dose that most male users have found is 12.5mg every other day.
Since Exemestane is so potent, most bodybuilders use a 12.5mg dose of Exemestane every other day since the half-life is 24 hours. 48 hours without another dose of Exemestane is still very sufficient to suppress Estrogen levels in the body.
EXEMESTANE CYCLE THERAPY
Exemestane is used as an On-Cycle Therapy (OCT) in very anabolic bodybuilding cycles like Testosterone, Deca, EQ, Dianabol, and others.
Assuming one knows the drug they’re using well and bloodwork has been done, Exemestane should be kept on-hand at all times to inhibit the conversion of Testosterone into Estrogen (Aromatization).
Exemestane is often a great substitute versus Anastrozole (Arimidex) due to less reported side-effects like depression, hot flashes, and weak bones.
EXEMESTANE IN BODYBUILDING
Bodybuilders will use Exemestane typically on an every other day basis. The normal dose is 12.5mg every other day but this can be increased to 25mg in situations of highly-dosed anabolics.
In a nutshell, we could say that Exemestane is a great and sometimes necessary addition to a cycle including Testosterone to prevent the conversion of excess Estrogen. Exemestane can synergistically stack with any highly aromatizing compound like Dianabol, Testosterone, or Deca.
WHERE TO BUY EXEMESTANE
If you’ve decided to research with Exemestane and want to find the best Exemestane for sale, choosing a reliable company to buy from is crucial, since buying it from a bad company could result in you getting no results or getting horrible side-effects due to being sold something that’s not actually Exemestane.
We’ve categorized two of our favorite vendors with two different administrations: liquid and capsule form Exemestane.
LIQUID EXEMESTANE: AMINO ASYLUM EXEMESTANE
For liquid Exemestane, We recommend going with Amino Asylum.
Key benefits of Amino Asylum:
- Competitive Prices
- One-Stop Shop
- Good Customer Support
- Fast Shipping
- High-Quality Products
- Easier product dosing (liquid is easier to manipulate)
Amino Asylum is our favorite SARMs and research chemical source on the market in 2022.
Amino Asylum is definitely one of the newer SARMs and research chemical companies on the block but they’re very quickly starting to build up a good reputation for their company, due to many customers giving raving reviews for their products.
You can buy Exemestane from them through the link below and use code ENHANCED20 to save 20% off your order
Here is the price with a 20% discount of Amino Asylum Exemestane for sale:
- Exemestane (Aromasin) 20mg/mL = $23.99
CAPSULE EXEMESTANE: SWISS CHEMS
If you’ve decided you don’t like liquid research chemicals, capsules are a safe option.
Capsule form Exemestane is just as effective as liquid Exemestane, however, it is a little harder to take less or more in this form (if one needed to).
For capsule Exemestane, we recommend Swiss Chems.
Here’s why we love Swiss Chems:
- Pharmacy Grade Products
- Third Party Tested For Purity
- Worldwide Shipping
- Competitive Prices
We asked for a coupon code to give you guys—use the code enhanced10 for 10% off. This will apply to any of the AI, PCT, SARM, or peptide that they’re selling on their site.
When you buy Exemestane from Swiss Chems, you’ll be provided with a third-party analysis of the batch purity of the drug you’re ordering for yourself
The product(s) will arrive at your doorstep the within days of you order. Plus, Swiss Chems backs it with a 30-day return guarantee and a 100% satisfaction guarantee.
Here is the price with a 10% discount of Swiss Chems Exemestane for sale:
- Exemestane (Aromasin) 12.5mg/cap = $69.25
Exemestane has a half-life of 24 hours.
Assuming one is taking it every other day or every two days, the blood levels would be closest to 0 around Day 4 after stopping Exemestane completely.
It's not expensive at Amino Asylum!
Research chemicals in general can be expensive, however, because of how well they work, how few the manufacturers are that produce them, and how even fewer their availability is with the sources that carry them.
Permanently deactivated aromatase enzymes.
Once the user stops Exemestane, many of the side-effects will subside.
The side-effects that won't go away immediately could be hormone-related effects like depression or lower bone density. All side-effects are reversible with other drugs, however.